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Design and synthesis of
pironetin analogues with simplified structure and study of their
interactions with microtubules.
J. A. Marco, J. García-Pla,
M. Carda, J. Murga, Eva Falomir, C. Trigili, S. Notararigo, J. F.
Díaz, I. Barasoain. Eur. J. Med.
Chem.
2011,
46, 1630-1637.
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Stereoselective
Synthesis of Five Biologically Active, Naturally Occurring Medium
and Large Ring Lactones.
J. A. Marco,
M. Carda. Nat. Prod. Commun.
2011, 6,
505-514.
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Synthesis and Biological
Properties of the Cytotoxic 14-Membered Macrolides Aspergillide A
and B. S. Díaz-Oltra, C. A.
Angulo-Pachón, J. Murga, E. Falomir, M. Carda, J. A. Marco.
Chem. Eur. J. 2011,
17, 675-688.
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Stereoselective Synthesis and
Structural Correction of the Naturally Occurring Lactone Stagonolide
G. C. A. Angulo-Pachón, S. Díaz-Oltra,
J. Murga, M. Carda, J. A. Marco.
Org.
Lett.
2010, 12, 5752-5755.
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The high affinity dopamine uptake inhibitor, JHW 007,
blocks cocaine-induced reward, locomotor stimulation and
sensitization.
C. Velázquez-Sánchez, A.
Ferragud, J. Murga, M. Carda, J. J. Canales.
European
Neuropsychopharmacology,
2010,
20, 501-508.
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Stereoselective synthesis
of the cytotoxic 14-membered macrolide aspergillide A.
S.
Díaz-Oltra, C. Angulo-Pachón, J. Murga, M. Carda, J.
A. Marco. J. Org. Chem.
2010, 75, 1775-1778.
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A formal, stereoselective synthesis of the natural
tetrahydropyran derivative ophiocerin D.
J. Paños, J. Murga, M. Carda, J. A. Marco.
Tetrahedron:Asymmetry
2010, 21, 425-428.
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Convergent, stereoselective
syntheses of the glycosidase inhibitors broussonetines C, O and P.
Celia Ribés, Eva Falomir, Juan Murga, Miguel Carda, J. Alberto Marco.
Tetrahedron
2009, 65, 10612-10616.
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A Dopamine Transport Inhibitor with Markedly Low
Abuse Liability Suppresses Cocaine Self-Administration in the Rat.
A.
Ferragud, C. Velázquez-Sánchez, V.
Hernández-Rabaza, A. Nácher, J. Murga, M. Carda, J. Canales.
Psychopharmacology 2009,
207, 281-289.
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The Dopamine Uptake Inhibitor
3a-[bis(40-fluorophenyl)metoxy]-tropane Reduces Cocaine-Induced
Early-Gene Expression, Locomotor Activity, and Conditioned Reward.
C.
Velázquez-Sánchez, A. Ferragud, V.
Hernández-Rabaza, A. Nácher, V.
Merino, M. Carda, J.
Murga, J. J.
Canales. Neuropsychopharmacology
2009,
34, 2497-2507.
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Stereoselective syntheses of
the glycosidase inhibitors hyacinthacine A2,
hyacinthacine A3 and 5-epi-hyacinthacine A3.
C. Ribes, E. Falomir, M. Carda, J. A. Marco.Tetrahedron
2009, 65, 6965-6971.
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Stereoselective synthesis of the cytotoxic
macrolide aspergillide B .
S. Díaz-Oltra,
C. A. Angulo-Pachón, M.
N. Kneeteman, J. Murga, M.
Carda, J. A. Marco.
Tetrahedron Lett.
2009, 50, 3783-3785.
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Convergent, stereoselective
syntheses of the glycosidase inhibitors broussonetines D and M.
C.
Ribes, E. Falomir, J.
Murga, M. Carda, J. A.
Marco. Org. Biomol. Chem.
2009, 7, 1355-1360.
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Stereoselective
Synthesis of the Naturally Occurring Pyrrolidine Radicamine B and a
Formal Synthesis of Nectrisine.
C. Ribes, E. Falomir, M. Carda, J.
A. Marco. J. Org. Chem.
2008, 73, 7779-7782.
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Double Diastereoselection in Aldol Reactions Mediated by
Dicyclohexylchloroborane between L-Erythrulose Derivatives and
Chiral α-Amino and α-Fluoro Aldehydes.
Relative Importance of Felkin-Anh and Cornforth
Transition States. S. Díaz-Oltra,
M. Carda, J. Murga, E. Falomir, J. A. Marco.
Chem. Eur. J.,
2008,
14, 9240-9254.
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Stereoselective Synthesis of the Naturally Occurring 2-Pyranone
Dodoneine.
P.
Álvarez-Bercedo, E. Falomir, J. Murga, M. Carda, J. A. Marco.
Eur. J. Org. Chem.,
2008 , 73, 4015-4018.
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Stereoselective
synthesis of the bacterial DNA primase inhibitor Sch 642305 and its
C-4 epimer. J.
García-Fortanet, M. Carda, A. Marco.
Tetrahedron 2007,
63, 12131-12137.
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The Total Synthesis and
Biological Properties of the Cytotoxic Macrolide FD-891 and its
Non-Natural (Z)-C12 Isomer.
J. García-Fortanet, J. Murga, M. Carda, J. A.
Marco, R. Matesanz, J. F. Díaz. I. Barasoaín.
Chem. Eur. J.,
2007,
13, 5060-5074.
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Stereoselective synthesis of
naturally occurring 5,6-dihydropyran-2-ones.
J. A. Marco, M. Carda, J.
Murga, y E. Falomir. Tetrahedron,
2007,
63, 2929-2958.
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Stereoselective synthesis of the glycosidase inhibitor australine
through a one-pot, double-cyclization strategy .
C. Ribes, E. Falomir, M. Carda y
J. A. Marco.
Org. Lett.
2007, 9, 77-80. -
Stereoselective synthesis of a C19-C26
fragment of amphidinolides
G and H. P. Formentín, J.
Murga, M. Carda y J. A. Marco. Tetrahedron:
Asymmetry,
2006,
17, 2938-2942.
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Enantioselective synthesis and absolute configurations of aculeatins
A, B, D, and 6-epi-aculeatin D.
P. Álvarez-Bercedo, E. Falomir, M. Carda y
J. A. Marco. Tetrahedron
2006, 62,
9641-9649.
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Stereoselective Synthesis of the Published
Structure of Feigrisolide A. Structural Revision of Feigrisolides A
and B.
P. Álvarez-Bercedo, J. Murga, M. Carda y
J. A. Marco. J. Org. Chem.
2006, 71,
5766-5769.
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Stereoselective Synthesis of the Cytotoxic
Macrolide FD-891. J. García-Fortanet,
J. Murga, M. Carda y J. A.
Marco. Org. Lett.
2006, 8,
2695-2698.
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The
Stereoselective Synthesis of the
Nonnatural Enantiomers of Communiols A-C.
A Stereochemical Correction.
J. Murga, E. Falomir, M. Carda y
J. A. Marco. Nat. Prod. Commun.
2006, 1, 237-245.
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Antiparasite and
antimycobacterial activity of passifloricin analogues.
W. Cardona, W. Quiñones,
S. Robledo, I. Darío Vélez, J. Murga, J. García-Fortanet, M. Carda,
D. Cardona y F. Echeverri.
Tetrahedron
2006, 62, 4086-4092.
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Selective cleavage of acetals with
ZnBr2 in dichlomethane. C.
Ribes, E. Falomir y J. Murga.
Tetrahedron
2006, 62, 1239-1244.
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Stereoselective Total Synthesis
and Absolute Configuration of the Natural Decanolides (-)-Microcarpalide
and (+)-Lethaloxin. The Identity of (+)-Lethaloxin and (+)-Pinolidoxin.
J. García-Fortanet, J. Murga, E. Falomir, M. Carda y
J. A. Marco.
J. Org.
Chem.
2005, 70, 9822-9827.
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Enantioselective synthesis and
absolute configurations of
aculeatins A and B. E.
Falomir, P. Álvarez-Bercedo,
M. Carda y J. A. Marco. Tetrahedron
Lett. 2005, 48, 8407-8410.
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Stereoselective
synthesis of
ent-communiols A-C.
J. Murga, E. Falomir,
M. Carda y J. A.
Marco. Tetrahedron Lett. 2005,
46, 8199-8202.
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Double
Diastereoselection in Aldol Reactions mediated by
Dicyclohexylchloroborane between Chiral Aldehydes
and A Chiral Ethyl Ketone Derived from L-Erythrulose
. S.
Díaz-Oltra, J. Murga, E. Falomir, M. Carda y J. A. Marco.
J. Org.
Chem.
2005, 70, 8130-8139.
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Stereoselective
addition of organometallic reagents to a chiral acyclic nitrone
derived from L-erythrulose. J. Murga,
R. Portolés, E. Falomir, M.
Carda y J. A. Marco.
Tetrahedron:
Asymmetry 2005,
16, 1807-1816.
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Stereoselective synthesis of the published structure of
synargentolide A and of one stereoisomer
thereof.
J. García-Fortanet, J. Murga,
M. Carda y J. A. Marco.
ARKIVOC 2005, part 9, 175-188.
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Stereoselective
Synthesis of the Naturally Occurring
Styryllactones (+)-Goniofufurone and (+)-Cardiobutanolide.
P. Ruiz, J. Murga, M. Carda y J. A. Marco.
J.
Org. Chem.
2005, 70, 713-716.
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Stereoselective
Synthesis of
the C1-C12 fragment of the cytotoxic macrolide
FD-891.
J. Murga, J. García-Fortanet,
M. Carda y J. A.
Marco. Synlett 2004, 2830-2832.
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Stereoselective
Synthesis of
hyptolide and 6-epi-hyptolide.
J. García-Fortanet, J.
Murga, M. Carda y
J.
A. Marco. Tetrahedron 2004,
60, 12261-12267.
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Stereoselective
Synthesis of the Antiprotozoal Lactone
Passifloricin A and Seven Isomers Thereof. J. Murga,
J. García-Fortanet, M.
Carda y J. A. Marco.
J. Org.
Chem.
2004, 69, 7277-7283.
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Stereoselective
Synthesis of
the C14-C26 fragment of the cytotoxic
macrolide FD-891.
J. Murga, J. García-Fortanet,
M. Carda y J. A.
Marco. Tetrahedron Lett. 2004,
45, 7499-7501.
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Stereoselective
Synthesis of Anamarine.
S. Díaz-Oltra, J. Murga, E. Falomir, M. Carda y J. A. Marco.
Tetrahedron
2004, 60, 2979-2985.
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Stereoselective anti Aldol reactions of
Erythrulose Derivatives. Functionalized Chiral d3 and d4
Synthons.
J. Murga, P. Ruiz, E. Falomir, M. Carda, G. Peris y J. A.
Marco.
J. Org.
Chem.
2004, 69, 1987-1992.
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Double
Diastereoselection in Aldol Reactions mediated by
Dicyclohexylchloroborane between Erythrulose Derivatives and Chiral
Aldehydes. The Felkin-Anh vs. Cornforth dichotomy
. J. A.
Marco, M. Carda, S. Díaz-Oltra, J. Murga, E. Falomir y H.
Röper.
J. Org.
Chem.
2003, 68, 8577-8582.
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Asymmetric Synthesis of
Passifloricin A: A Correction in Structure.
J. Murga, J. García-Fortanet,
M. Carda y J. A.
Marco. Tetrahedron Lett. 2003,
44, 7909-7912.
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Stereoselective
Synthesis and Determination of the Cytotoxic Properties of
Spicigerolide and Three of Its Stereoisomers.
E. Falomir, J. Murga, P. Ruiz, M. Carda, J. A. Marco, R.
Pereda-Miranda, M. Fragoso-Serrano y C. M. Cerda-García-Rojas.
J.
Org. Chem.
2003, 68,
5672-5676.
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On the Structure of Passifloricin A:
Asymmetric Synthesis of the d-Lactones of (2Z,5S,7R,9S,11S)- and
(2Z,5R,7R,9S,11S)-Tetrahydroxyhexacos-2-enoic Acid.
J. García-Fortanet, J.
Murga, M. Carda, J. A. Marco. Org. Lett.
2003,
10 , 1447-1449.
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Stereoselective synthesis of (+)-hyptolide. J. Murga, J. García-Fortanet,
M. Carda, J. A. Marco. Tetrahedron Lett. 2003, 44,
1737-1739.
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Stereoselective
synthesis of spicigerolide. E. Falomir,
J. Murga, M. Carda y J. A. Marco. Tetrahedron
Lett. 2003, 44, 539-541.
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Stereoselective synthesis of (-)-maliyngolide, (+)-malyngolide and
(+)-tanikolide using ring-closing metathesis. M. Carda, S.
Rodríguez, E. Castillo, A. Bellido, S. Díaz-Oltra y J. A. Marco.
Tetrahedron 2003, 59, 857-864.
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Erythrulose derivatives as functionalized
chiral d3 and d4 synthons.
J. Murga, E. Falomir, M. Carda y J. A. Marco.
Tetrahedron Asymmetry 2002, 13 , 2317-2327.
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Influence of the Protecting Groups on the syn/anti Stereoselectivity
of Boron Aldol Additions with Erythrulose Derivatives. A Theoretical
and Experimental Study.
J. Murga, E. Falomir, F. González, M. Carda y J. A. Marco.
Tetrahedron 2002, 58 , 9697-9707.
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Stereoselective síntesis of
microcarpalide. J. Murga, E. Falomir,. J.
Garcia-Fortanet, M. Carda y J. A. Marco. Org.
Lett. 2002, 4 , 3447-3449.
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Stereoselective
synthesis of the naturally occurring lactones (-)-osmundalactone and
(-)-muricatacine using ring-closing metathesis.
M. Carda, S.
Rodríguez, F. González, E. Castillo, A. Villanueva, J. A. Marco.
Eur. J.
Org. Chem.
2002, 2649-2655.
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Stereoselective
synthesis of (-)-cytoxazone.
M. Carda, F.
González, R. Sánchez, J. A. Marco.
Tetrahedron: Asymmetry
2002, 13, 1005-1010.
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Stereoselective
Synthesis of (+)-Boronolide.
M. Carda, S.
Rodríguez, B. Segovia, J. A. Marco.
J. Org.
Chem.
2002, 67, 6560-6563.
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Synthesis of a,a-disubstituted a-amino acid
derivatives in enantiopure form via stereoselective addition of
Grignard reagents to a chiral acyclic nitrone derived from L-erythrulose.
R. Portolés, J. Murga, E. Falomir, M. Carda, S. Uriel y J. A.
Marco. Synlett 2002, 711-714.
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Synthesis of Conjugated
d-Lactams
Using Ring-Closing Metathesis.
S.
Rodríguez, E. Castillo, M. Carda, J. A. Marco.
Tetrahedron
2002,
58,
1185-1192.
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Stereoselective Allylations of Erythrulose Derivatives Under
Anhydrous Conditions.
M. Carda, E.
Castillo, S. Rodríguez, F. González, J. A. Marco.
Tetrahedron: Asymmetry
2001, 12,
1417-1429.
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An ab initio Study of the Enolboration of
3-Pentanone Mediated by Boron Monochlorides L2BCl.
J. Murga, E. Falomir, M. Carda y J. A. Marco.
Tetrahedron 2001, 57, 6239-6247.
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Chlorodicyclohexylborane-Mediated Aldol
Additions of a,a´-Dioxygenated Ketones.
J. Murga, E. Falomir, M. Carda, F.
González y J. A. Marco.
Org.
Lett.
2001, 3,
901-904.
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Stereoselective
1,3-Dipolar Cycloadditions of a Chiral Nitrone Derived from
Erythrulose. An Experimental and DFT Theoretical Study.
M.
Carda, R.
Portolés, J.
Murga, S. Uriel,
J. A. Marco, L.
R. Domingo, R. J.
Zaragozá y H.
Röper. J. Org. Chem. 2000,
65, 7000-7009.
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Stereoselective Synthesis of syn-a-methyl-b-hydroxy
Esters.
M. Carda, J. Murga, E. Falomir, F. González y
J. A. Marco. Tetrahedron Asymmetry 2000,
11, 3211-3220.
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A
stereoselective synthesis of (+)-malyngolide via a ring-closing
olefin metathesis.
M. Carda ,
E. Castillo, S. Rodríguez, J. A. Marco.
Tetrahedron Lett. 2000, 41, 5511-5513.
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Aldol reactions with Erytrulose Derivatives:
Stereoselective Synthesis of Differentially Protected syn-a-b-Dihydroxy
Esters .
M. Carda, J. Murga, E. Falomir, F.
González y J. A. Marco.
Tetrahedron 2000,
56, 677-683.
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